SPYRAKIS, FRANCESCA
SPYRAKIS, FRANCESCA
SCIENZA E TECNOLOGIA DEL FARMACO
Application of an in house bioisosteric approach to the design of innovative inhibitors of aldo-keto reductase 1C3 (AKR1C3)
2019-01-01 Chiara Vigato, Agnese Chiara Pippione, Sandra Kovachka, Francesca Spyrakis, Martina Daga, Simonetta Oliaro-Bosso, Marco Lucio Lolli, Donatella Boschi
Application of an in house bioisosteric approach to the design of innovative inhibitors of aldo-keto reductase 1C3 (AKR1C3)
2019-01-01 Chiara Vigato, Agnese Chiara Pippione, Sandra Kovachka, Francesca Spyrakis, Martina Daga, Simonetta Oliaro Bosso, Marco Lucio Lolli, Donatella Boschi
BROAD SPECTRUM METALLO beta-LACTAMASES INHIBITORS: NEW TOOLS AGAINST CLINICALLY-RELEVANT CARBAPENEMASES
2022-01-01 Lazzarato, L.; Failla, M.; Gianquinto, E.; Bersani, M.; Bertarini, L.; Verri, A.; Vascon, F.; Sannio, F.; Verdirosa, F.; Beatrice, N.; De Luca, F.; Costi, M.P.; Cruciani, G.; Docquier, J.D.; Cendron, L.; Spyrakis, F.; Tondi, D.
In the search for new NLRP3 inhibitors: chemical modulation of the 1-(piperidin-4-yl)-1,3-dihydro-2 Hbenzo[d]imidazole-2-one scaffold
2021-01-01 Simone Gastaldi, Valentina Boscaro, Eleonora Gianquinto, Christina F. Sandall, Marta Giorgis, Elisabetta Marini, Federica Blua, Margherita Gallicchio, Francesca Spyrakis, Justin A. MacDonald, Massimo Bertinaria
Indomethacin Inhibits Proliferation In Cells Harbouring PIK3CA Mutations
2017-01-01 M. Gallicchio, M. Lolli, F. Spyrakis, D. Bonanni, V. Boscaro
Multiple-targeting ligands for AKR1C3 enzyme and androgen receptor to target prostate cancer
2021-01-01 Agnese Chiara Pippione, Zuhal Kilic-Kurt, Stefano Sainas, Iole Mannella, Barbara Rolando, Sandra Kovachka, Francesca Spyrakis, Annamaria Buschini, Serena Montalbano, Simonetta Oliaro Bosso, Marco Lolli, Donatella Boschi
New Hydroxybenzoazole Inhibitors of Aldo-Keto Reductase 1C3 (AKR1C3): Disclosure of SAR Investigation to Target Prostate Cancer
2022-01-01 Chiara Vigato, Agnese Chiara Pippione, Iole Mannella, Mariia Iakovleva, Stefano Sainas, Simonetta Oliaro Bosso, Barbara Rolando, Sandra Kovachka, Francesca Spyrakis, Marco Lucio Lolli, Donatella Boschi
New inhibitors of Aldo-Keto Reductase 1C3 (AKR1C3) based on benzoisoxazole scaffold and their potential application in cancer
2021-01-01 Mannella, Iole, Vigato, Chiara, Pasha, Rabia; Pippione Agnese Chiara, Sainas, Stefano, Oliaro Bosso Simonetta; Rolando, Barbara; Kovachka, Sandra, Spyrakis, Francesca; Boschi, Donatella, Lolli. Marco Lucio
Strigolactone analogs are promising antiviral agents against Herpesviruses
2021-01-01 Matteo Biolatti, Marco Blangetti, Giulia D’Arrigo, Francesca Spyrakis, Paola Cappello, Camilla Albano, Sergio Fernando Castillo Pacheco, Santo Landolfo, Cristina Prandi, Marco De Andrea, Valentina Dell’Oste
Strigolactone Analogs Are Promising Antiviral Agents for the Treatment of Human Cytomegalovirus Infection
2020-01-01 CAMILLA ALBANO, MATTEO BIOLATTI, MARCO BLANGETTI, GIULIA D’ARRIGO, FRANCESCA SPYRAKIS, PAOLA CAPPELLO, PAOLO RAVANINI, SELINA PASQUERO, FRANCESCA GUGLIESI, SERGIO F. CASTILLO PACHECO, SANTO LANDOLFO, MARCO DE ANDREA, CRISTINA PRANDI, VALENTINA DELL’OSTE
Strigolactone analogs are promising antiviral agents for the treatment of human cytomegalovirus infection
2021-01-01 MATTEO BIOLATTI , MARCO BLANGETTI , GIULIA D’ARRIGO, FRANCESCA SPYRAKIS, PAOLA CAPPELLO, CAMILLA ALBANO, SERGIO FERNANDO CASTILLO PACHECO, LINDA TRIFIRO’ , PAOLO RAVANINI , SANTO LANDOLFO, MARCO DE ANDREA, CRISTINA PRANDI , VALENTINA DELL’OSTE
Strigolactones as antiviral drugs to inhibit Herpesvirus replication
2019-01-01 SELINA PASQUERO, GLORIA GRIFFANTE, FRANCESCA GUGLIESI, VALENTINA DELL’OSTE, MATTEO BIOLATTI, GANNA GALITSKA, MARCO BLANGETTI, CRISTINA PRANDI, PAOLA CAPPELLO, FRANCESCA SPYRAKIS, GIULIA D’ARRIGO, MARCO DE ANDREA, SANTO LANDOLFO
Strigolactones as broad-spectrum antivirals against β-coronaviruses through targeting SARS-CoV-2 Mpro
2022-01-01 Camilla Albano, Matteo Biolatti, Marco Blangetti, Greta Bajetto, Davide Arnodo, Melissa Baggeri, Matteo Bersani, Giulia D’Arrigo, Marco De Andrea, Francesca Gugliesi, Selina Pasquero, Ivan Visentin, Cristina Prandi, Francesca Spyrakis, Fabio Magurano, Valentina Dell’Oste
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Application of an in house bioisosteric approach to the design of innovative inhibitors of aldo-keto reductase 1C3 (AKR1C3) | 2019 | Chiara Vigato, Agnese Chiara Pippione, Sandra Kovachka, Francesca Spyrakis, Martina Daga, Simonetta Oliaro-Bosso, Marco Lucio Lolli, Donatella Boschi | |
Application of an in house bioisosteric approach to the design of innovative inhibitors of aldo-keto reductase 1C3 (AKR1C3) | 2019 | Chiara Vigato, Agnese Chiara Pippione, Sandra Kovachka, Francesca Spyrakis, Martina Daga, Simonetta Oliaro Bosso, Marco Lucio Lolli, Donatella Boschi | |
BROAD SPECTRUM METALLO beta-LACTAMASES INHIBITORS: NEW TOOLS AGAINST CLINICALLY-RELEVANT CARBAPENEMASES | 2022 | Lazzarato, L.; Failla, M.; Gianquinto, E.; Bersani, M.; Bertarini, L.; Verri, A.; Vascon, F.; Sannio, F.; Verdirosa, F.; Beatrice, N.; De Luca, F.; Costi, M.P.; Cruciani, G.; Docquier, J.D.; Cendron, L.; Spyrakis, F.; Tondi, D. | |
In the search for new NLRP3 inhibitors: chemical modulation of the 1-(piperidin-4-yl)-1,3-dihydro-2 Hbenzo[d]imidazole-2-one scaffold | 2021 | Simone Gastaldi, Valentina Boscaro, Eleonora Gianquinto, Christina F. Sandall, Marta Giorgis, Elisabetta Marini, Federica Blua, Margherita Gallicchio, Francesca Spyrakis, Justin A. MacDonald, Massimo Bertinaria | |
Indomethacin Inhibits Proliferation In Cells Harbouring PIK3CA Mutations | 2017 | M. Gallicchio, M. Lolli, F. Spyrakis, D. Bonanni, V. Boscaro | |
Multiple-targeting ligands for AKR1C3 enzyme and androgen receptor to target prostate cancer | 2021 | Agnese Chiara Pippione, Zuhal Kilic-Kurt, Stefano Sainas, Iole Mannella, Barbara Rolando, Sandra Kovachka, Francesca Spyrakis, Annamaria Buschini, Serena Montalbano, Simonetta Oliaro Bosso, Marco Lolli, Donatella Boschi | |
New Hydroxybenzoazole Inhibitors of Aldo-Keto Reductase 1C3 (AKR1C3): Disclosure of SAR Investigation to Target Prostate Cancer | 2022 | Chiara Vigato, Agnese Chiara Pippione, Iole Mannella, Mariia Iakovleva, Stefano Sainas, Simonetta Oliaro Bosso, Barbara Rolando, Sandra Kovachka, Francesca Spyrakis, Marco Lucio Lolli, Donatella Boschi | |
New inhibitors of Aldo-Keto Reductase 1C3 (AKR1C3) based on benzoisoxazole scaffold and their potential application in cancer | 2021 | Mannella, Iole, Vigato, Chiara, Pasha, Rabia; Pippione Agnese Chiara, Sainas, Stefano, Oliaro Bosso Simonetta; Rolando, Barbara; Kovachka, Sandra, Spyrakis, Francesca; Boschi, Donatella, Lolli. Marco Lucio | |
Strigolactone analogs are promising antiviral agents against Herpesviruses | 2021 | Matteo Biolatti, Marco Blangetti, Giulia D’Arrigo, Francesca Spyrakis, Paola Cappello, Camilla Albano, Sergio Fernando Castillo Pacheco, Santo Landolfo, Cristina Prandi, Marco De Andrea, Valentina Dell’Oste | |
Strigolactone Analogs Are Promising Antiviral Agents for the Treatment of Human Cytomegalovirus Infection | 2020 | CAMILLA ALBANO, MATTEO BIOLATTI, MARCO BLANGETTI, GIULIA D’ARRIGO, FRANCESCA SPYRAKIS, PAOLA CAPPELLO, PAOLO RAVANINI, SELINA PASQUERO, FRANCESCA GUGLIESI, SERGIO F. CASTILLO PACHECO, SANTO LANDOLFO, MARCO DE ANDREA, CRISTINA PRANDI, VALENTINA DELL’OSTE | |
Strigolactone analogs are promising antiviral agents for the treatment of human cytomegalovirus infection | 2021 | MATTEO BIOLATTI , MARCO BLANGETTI , GIULIA D’ARRIGO, FRANCESCA SPYRAKIS, PAOLA CAPPELLO, CAMILLA ALBANO, SERGIO FERNANDO CASTILLO PACHECO, LINDA TRIFIRO’ , PAOLO RAVANINI , SANTO LANDOLFO, MARCO DE ANDREA, CRISTINA PRANDI , VALENTINA DELL’OSTE | |
Strigolactones as antiviral drugs to inhibit Herpesvirus replication | 2019 | SELINA PASQUERO, GLORIA GRIFFANTE, FRANCESCA GUGLIESI, VALENTINA DELL’OSTE, MATTEO BIOLATTI, GANNA GALITSKA, MARCO BLANGETTI, CRISTINA PRANDI, PAOLA CAPPELLO, FRANCESCA SPYRAKIS, GIULIA D’ARRIGO, MARCO DE ANDREA, SANTO LANDOLFO | |
Strigolactones as broad-spectrum antivirals against β-coronaviruses through targeting SARS-CoV-2 Mpro | 2022 | Camilla Albano, Matteo Biolatti, Marco Blangetti, Greta Bajetto, Davide Arnodo, Melissa Baggeri, Matteo Bersani, Giulia D’Arrigo, Marco De Andrea, Francesca Gugliesi, Selina Pasquero, Ivan Visentin, Cristina Prandi, Francesca Spyrakis, Fabio Magurano, Valentina Dell’Oste |